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LEDアレーシステム使用研究論文リスト

当社のLEDアレーシステムを使用した論文のリストです。論文の内容を示すキーワードを併記しております。キーワードをクリックするとキーワードが一致する論文のリストが表示されます。

キーワードリスト

Photoswitchable positive allosteric modulators of metabotropic glutamate receptor 4 to improve selectivity

Silvia Panarello, Aleix González-Díez, Alice E. Berizzi, Fanny Malhaire Roser Borràs-Tudurí Xavier Rovira Carme Serra Laurent Prézeau Jean-Philippe Pin Cyril Goudet Amadeu Llebaria Xavier Gómez-Santacana

iScience. 2024 May 28. https://doi.org/10.1016/j.bcp.2024.116396

A high-affinity, cis-on photoswitchable beta blocker to optically control β2-adrenergic receptors in vitro and in vivo

Shuang Shi, Yang Zheng, Joëlle Goulding, Silvia Marri, Laura Lucarini, Benjamin Konecny, Silvia Sgambellone, Serafina Villano, Reggie Bosma, Maikel Wijtmans, Stephen J. Briddon, Barbara A. Zarzycka, Henry F. Vischer, Rob Leurs

Biochem. Pharmacol. 2024 June 26. https://doi.org/10.1016/j.isci.2024.110123

Crystal structure reveals the binding mode and selectivity of a photoswitchable ligand for the adenosine A2A receptor

Tsuyoshi Araya, Yuya Matsuba, Harufumi Suzuki, Tomohiro Doura, Nipawan Nuemket, Eriko Nango, Masaki Yamamoto, Dohyun Im, Hidetsugu Asada, Shigeki Kiyonaka, So Iwata

Biochem Biophys Res Commun . 2024 Feb 5:695:149393. doi: 10.1016/j.bbrc.2023.149393.

Optogluram-2: a subtype-selective photoswitchable positive allosteric modulator for metabotropic glutamate receptor 4

Silvia Panarello, Aleix González-Díez, Alice Berizzi, Fanny Malhaire, Roser Borràs-Tudurí, Xavier Rovira, Laurent Prezeau, Jean-Philippe Pin, Cyril Goudet, Amadeu Llebaria, Xavier Gómez-Santacana

Authorea. July 03, 2023. DOI: 10.22541/au.168837491.17051077/v1

Visible-Light-Controlled Histone Deacetylase Inhibitors for Targeted Cancer Therapy

Laia Josa-Culleré, Amadeu Llebaria

J Med Chem. 2023 Jan 18. doi: 10.1021/acs.jmedchem.2c01713

Design and development of photoswitchable DFG-Out RET kinase inhibitors

Yongjin Xu, Chunxia Gao, Måns Andreasson, Liliana Håversen, Marta P Carrasco, Cassandra Fleming, Thomas Lundbäck, Joakim Andréasson, Morten Grøtli

Eur J Med Chem . 2022 Mar 10;234:114226. doi: 10.1016/j.ejmech.2022.114226

Agonists and allosteric modulators promote signaling from different metabotropic glutamate receptor 5 conformations

Chady Nasrallah, Giuseppe Cannone, Julie Briot, Karine Rottier, Alice E Berizzi, Chia-Ying Huang, Robert B Quast, Francois Hoh, Jean-Louis Banères, Fanny Malhaire, Ludovic Berto, Anaëlle Dumazer, Joan Font-Ingles, Xavier Gómez-Santacana, Juanlo Catena, Julie Kniazeff, Cyril Goudet, Amadeu Llebaria, Jean-Philippe Pin, Kutti R Vinothkumar, Guillaume Lebon

Cell Rep . 2021 Aug 31;36(9):109648. doi: 10.1016/j.celrep.2021.109648.

Mechanistic insights into light-driven allosteric control of GPCR biological activity

Maria Ricart Ortega , Alice E. Berizzi, Vanessa Pereira, Fanny Malhaire, Juanlo Catena, Joan Font, Xavier Gomez-Santacana, Lourdes Muñoz, Charleine Zussy, Carmen Serra, xavier Rovira, Cyril Goudet, and Amadeu Llebaria

ACS Pharmacol. Transl. Sci. 2020Aug DOI: 10.1021/acsptsci.0c00054

Photoswitchable Antagonists for a Precise Spatiotemporal Control of β2-Adrenoceptors

Anna Duran-Corbera , Juanlo Catena, Marta Otero-Viñas, Amadeu Llebaria, Xavier Rovira

J. Med. Chem. 2020, 63, 15, 8458-8470 DOI: 10.1021/acs.jmedchem.0c00831